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International Symposium on Chemistry, Biology and Medicine |
Program schedule (20/04/2006 - 58 KB)
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28/05/2006 |
14:00 | Registration |
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18:00 | Welcome Reception |
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19:00 | Live Performance of Cypriot and Greek Songs by the Choir of Karavas Organization |
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29/05/2006 |
08:00 | Welcome and Opening remarks |
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08:40 | Natural Product Synthesis: A Stimulus for Discovery |
Prof. Steven V. LEY (UNIVERSITY OF CAMBRIDGE, Cambridge, United Kingdom) |
09:30 | Coffee break and Poster session |
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10:00 | Multidimensional Lead Optimization: The Discovery of Innovative Small Molecule Therapeutics |
Prof Magid ABOU-GHARBIA (TEMPLE UNIVERSITY, Philadelphia, United States) |
10:50 | Reactivity and Applications of a New Diene for Organic Synthesis |
Prof. Erik SORENSEN (PRINCETON UNIVERSITY, Princeton, United States) |
11:30 | The Discovery of Non Transition-State Isostere BACE Inhibitors |
Dr Philippe NANTERMET (MERCK AND CO., WEST POINT, United States) |
12:00 | Lunch and Poster session |
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14:00 | Mini Business Symposium and Panel Discussion |
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14:01 | Chemistry in Drug Discovery: New Trends and New Challenges.
Coordinator: Dr Ron Magolda, Wyeth Research, Princton, USA.
Participants: to be announced |
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14:02 | New Trends in Chemistry Outsourcing.
Coordinator: Dr Eugene Vaisberg, ChemBridge, San Diego, USA.
Participants: to be announced |
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30/05/2006 |
08:00 | Synthetic Investigations of Antimitotic Agents |
Prof. Madeleine JOULLIÉ (UNIVERSITY OF PENNSYLVANIA, Philadelphia, United States) |
08:50 | From Chemistry to Medicine: New Chemical Reactions and New Synthetic Molecules Leading to New Therapies for Inflammation and Cancer |
Prof. Nicos A. PETASIS (UNIVERSITY OF SOUTHERN CALIFORNIA, LOS ANGELES, United States) |
09:30 | Coffee break and Poster session |
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10:00 | Structure-based Design of Nuclear Receptor Hormone Ligands: Potent Quinoline-based Liver X Receptor (LXR) Agonists
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Dr Ronald MAGOLDA (WYETH RESEARCH, Monmouth Junction,, United States) |
10:30 | TAFIa Inhibitors for Treatment of Thrombosis |
Dr Mark BUNNAGE (PFIZER, Boston, United States) |
11:00 | From the Insoluble Dye Indirubin Towards Highly Active, Soluble
CDK2-Inhibitors |
Dr Rolf JAUTELAT (SCHERING, Berlin, Germany) |
11:30 | Discovery of Pyrido-Pyrimidone Based Selective and Orally Efficacious p38 MAP Kinase Inhibitors |
Dr Swaminathan (Ravi) NATARAJAN (MERCK, Rahway, United States) |
12:00 | Lunch and Poster session |
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14:00 | A Multi-dimensional Approach to Molecular Recognition in Chemistry and Biology: Towards New Antimalarial Therapies |
Prof. François DIEDERICH (ETH ZURICH, Zürich, Switzerland) |
14:50 | Towards Measuring and Modulating Protein Function with Small Molecules |
Prof. Nicolas WINSSINGER (UNIVERSITY OF STRASBOURG, Strasbourg, France) |
15:30 | Coffee break |
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15:50 | Discovery and Optimization of Novel Drug Like Molecules via the ConTourTM Design Technology |
Dr David CLAREMON (VITAE PHARMACEUTICAL, Fort Washington, United States) |
16:20 | Development of Transition Metal Catalyzed Reaction for Organic Synthesis |
Prof. F. Dean TOSTE (UNIVERSITY OF CALIFORNIA, Berkeley, United States) |
31/05/2006 |
08:00 | Structure-based Organic Synthesis of Drug Prototypes |
Prof. Stephen HANESSIAN (UNIVERSITY OF MONTREAL, MONTREAL, QC, Canada) |
08:50 | Chemistry and Biology of Heterocycles: From Combinatorial Chemistry to Natural Product Synthesis |
Prof. Stefan BRAESE (UNIVERSITY OF KARLSRUHE, KARLSRUHE, Germany) |
09:30 | Coffee break and Poster session |
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10:00 | Stereoselective Synthesis of Biologically Active Alkaloids |
Prof. David TANNER (THE TECHNICAL UNIVERSITY OF DENMARK, LYNGBY, Denmark) |
10:40 | Geometric Control of Alkenes in Organic Synthesis |
Prof. Jun'ichi UENISHI (KYOTO PHARMACEUTICAL UNIVERSITY, KYOTO, Japan) |
11:20 | Natural Products; Targets of Opportunities |
Prof. Emmanuel THEODORAKIS (UNIVERSITY OF CALIFORNIA SAN DIEGO, La Jolla, United States) |
12:00 | Lunch and Poster session |
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14:00 | Excursion
Details to be announced |
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19:00 | Nicolaou Group Re-union Dinner |
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01/06/2006 |
08:00 | Melatonin, a Hormone in the Dark |
Prof. Peter J. GARRATT (UNIVERSITY COLLEGE LONDON, London, United Kingdom) |
08:50 | Synthesis Adventures with Bases and Bridges |
Prof. Nigel SIMPKINS (UNIVERSITY OF NOTTINGHAM, NOTTINGHAM, United Kingdom) |
09:30 | Coffee break an dPoster session |
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10:00 | Biocatalysis: Key Element in the Synthesis of Bioactive Heterocycles and Natural Products |
Prof. Floris RUTJES (RADBOUD UNIVERSITY NIJMEGEN, Nijmegen, The Netherlands) |
10:40 | Study towards the Total Synthesis of Micrandilactone A |
Prof. Zhen YANG (PEKING UNIVERSITY, BOSTON, United States) |
11:20 | Inhibition of the Formation of the Transcription Activation Complex by the Thyroid Hormone Receptor |
Dr Rodney KIP GUY (ST. JUDE CHILDREN'S RESEARCH HOSPITAL, Memphis, United States) |
12:00 | Lunch and Poster session |
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14:00 | Asymmetric Two-Center Catalysis: Construction of Tetrasubstituted Carbons |
Prof. Masakatsu SHIBASAKI (UNIVERSITY OF TOKYO, Tokyo, Japan) |
14:50 | The Catalytic Cycle of Discovery in Total Synthesis |
Prof. Phil BARAN (SCRIPPS RESEARCH INSTITUTE, La Jolla, United States) |
15:30 | Coffee break |
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16:40 | The Art of Total Synthesis at the Limits of Chemical Complexity |
Prof. K.C. NICOLAOU (THE SCRIPPS RESEARCH INSTITUTE, Houston, United States) |
17:00 | Closing |
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19:00 | Banquet |
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