ECHC 08 - XXIIIrd European Colloquium on Heterocyclic Chemistry 09/09/2008
Chairman
Dr Lieven MEERPOEL
19:00 Evening lecture on the life, work and personality of Dr. P. Janssen (founder of Janssen Pharmaceutica).
Dr. Paul J. LEWI
10/09/2008
08:45 Opening Ceremony
Chairman
Prof. Mikael BEGTRUP
09:00 Synthesis of Heterocycles via Alkoxyallenes
Prof. Hans-Ulrich REISSIG
09:50 JNJ-26483327 - A 'Macrocyclic' Multi-Targeted Kinase Inhibitor in Phase I Clinical Trials for the Treatment of Cancer
Dr. Eddy FREYNE
10:20 Ring Transformations and Peculiar Reactions of Functionalized β-Lactams
Prof. Norbert DE KIMPE
11:10 Coffee
11:40 Oral Communications - Session 1
Chairmen
Dr. Koen VAN AKEN (ECOSYNTH, Oostende, Belgium) Prof. Christian STEVENS (UGENT, Ghent, Belgium) Prof. Kourosch ABBASPOUR TEHRANI (VUB, Antwerp, Belgium)
(R1) (R2) (R3)
Synthesis and Cytotoxicity Evaluation of New Aziridine Containing Benzimidazolequinones
Dr. Fawaz ALDABBAGH
Addition of Organometallics to Cyclic Nitrones: Key Step for the Synthesis of Potent Inhibitors of Alpha-L-Fucosidases
Ms Amélie CASTIGLIA
Application of Microwave-Irradiation as Efficient and Green Reaction Conditions for Various Cycloadditions of 2H -Pyran-2-ones
Dr Kristof KRANJC
Synthesis and Properties of New Fluorophores with a Pyrimidine Central Unit
Prof Georges DUPAS
Synthesis of New Pyrimido[5,4-d ]Pyrimidinones
Dr Ana Helena BACELAR
Transformations of 3,3-Dichloroazetidines to Alkynylimines via 3-Chloro-2-azetines as Strained Intermediates
Dr Sven MANGELINCKX
Novel Routes towards Arylated Oxazoles and Thiazoles through Regioselective Direct C-H Arylation of Oxazole and Thiazole 4-carboxylate Scaffolds
Dr Christophe HOARAU
Preparation, Structural Studies and Reactivity of 1,2-Diazetidines
Mr Mike BROWN
Functionalized 2,5-Diryridinyl-pyrroles by Electrochemical Reduction of 3,6-Dipyridinyl-pyridazine Precursors
Ms Cécile MARIE
12:35 Lunch
13:20 Poster Session 1
Chairman
Prof. Gyorgy HAJÓS
14:20 Novel Organometallic Routes to Polyheterocyclic Ring Systems of Pharmacological Interest
Prof. Hans-Joachim KNÖLKER
14:50 Versatile Synthesis of Novel Ring-Fused 1,5-Benzodiazepines
Dr. Koen VANDYCK
15:20 Competitive Rearrangements of O-N Bond Containing Azoles: the "Power" of a "Weak" Bond
Prof. Andrea PACE
15:50 Coffee
Chairman
Prof. Dirk TOURWE
16:20 Applications of 3-Amino-2-Piperidones to the Synthesis of Peptidomimetics
Prof. Anna DIEZ
16:50 Making and Breaking Heterocyclic Rings via Metal Catalyzed Reactions
Prof. Mark LAUTENS
17:50 Transportation to the City
20:00 Concert in the Cathedral
11/09/2008
Chairman
Prof. Branko STANOVNIK
09:00 Organocatalytic versus Metal-Catalysed Selective Indole Functionalisation: Just a Matter of Choice?
Prof. Alfredo RICCI
09:50 Novel Synthesis of 2,4-Disubstituted Pyrimidines, Key Intermediates in the Synthesis of HIV Compounds
Dr. Fred STAPPERS
10:20 Synthesis and Properties of Novel (Indolo)carbazole Materials
Prof. Wim DEHAEN
11:10 Coffee
11:40 Oral Communications - Session 2
Chairmen
Prof. Kourosch ABBASPOUR TEHRANI (VUB, Antwerp, Belgium) Dr. Koen VAN AKEN (ECOSYNTH, Oostende, Belgium) Dr Pieter VAN DER VEKEN (UNIVERSITY OF ANTWERP, Antwerpen, Belgium)
(R1) (R2) (R3)
A New Synthesis of Substituted Pyrrole-2-Carboxylates by a Tandem Sonogashira Coupling 5-Endo-DIG-Cyclization from a beta-Iododehydrophenylalanine and Terminal Alkynes
Dr Agathe BEGOUIN
New Meso-Tetraarylporphyrin Derivatives via N-H Insertion Reactions with Diazo Compounds
Ms Ana Teresa PEIXOTO DE CAMPOS GOMES
Functional Analogues of Tröger's Base: New Synthetic Methods and Facile, Predictable Chromatographic Means for the Separation of Enantiomers
A Regio- and Stereospecific Synthesis of t -4-Amino-3-hydroxy- and t ,t -4-Amino-3,5-dihydroxypiperidines
Dr Igor TRUSHKOV
A Novel Multicomponent Reaction towards Imidazolidine-2-thions
Mr Maurice MOOIJMAN
A Novel Practical Synthesis of Licofelone
Prof. Stanislav RADL
Sequential Metal-Catalyzed N-Heteroarylation and C–C Cross-Coupling Reactions: An Expedient Route to Tris (hetero)aryl Systems
Mr Jamie SIDDLE
Toward the Total Synthesis of Enantiomerically Pure Antitumor Agent : TMC-69-6H
Ms Sophie VUONG
Polynitrogen Fused Tricyclic Compounds via a Nitrene-Mediated N-N Bond Formation
Ms Coralie NYFFENEGGER
Monocyclic and Dimeric 1,2,4-Triazines Useful Substrates for the Preparation of New Heterocyclic Systems and Natural Products
Dr Andrzej RYKOWSKI
3+2 Cycloadditions of 3-Pyrazolidinone-1-azomethine Imines: an Easy Access to Polysubstituted Pyrazolo[1,2-a ]pyrazolones
Prof. Jurij SVETE
An Efficient Microwave-Assisted Synthesis of Disubstituted 2-Amino-1H -imidazoles
Mr Denis ERMOLATEV
12:55 Lunch
13:40 Poster Session 2
Chairman
Prof. Johan VAN DER EYCKEN
14:40 Recent Developments Employing Heterocycles in Asymmetric Catalysis
Prof. Patrick GUIRY
15:10 Pyrrolidinones and Oxindoles as Templates for the Discovery of Innovative Treatments of Epilepsy
Dr. Laurent TURET
15:40 New Catalytic Reactions Designed for the Efficient Synthesis of Natural Products
Prof. Timothy DONOHOE
16:10 Coffee
Chairman
Prof. Guy QUÉGUINER
16:40 Palladium-Catalyzed Multicomponent and Domino Processes for Syntheses of Heterocycles
Prof. Jieping ZHU
17:10 Quinolones, Bisquinolones and Microwaves
Prof. Oliver KAPPE
18:00 Transportation to the City
12/09/2008
Chairman
Prof. Volker JÄGER
09:00 Selective Introduction of a Nitrogen-Containing Functionality into Organic Molecules
Prof. Slovenko POLANC
09:50 Golden Tools for the Synthesis of Heterocycles
Prof. Stephen HASHMI
10:20 Conferences Announcements
Chairman
Prof. Henk VAN DER PLAS
10:30 SNH Reactions in Heterocycles
Prof. Oleg CHUPAKHIN
11:20 Coffee
Chairman
Dr Laurent PROVINS
11:50 Novel Indole Chemistry in the Synthesis of Heterocycles
Prof. Gordon GRIBBLE
12:20 Efficient Synthesis of Heterocyclic Natural Products and Materials by Domino Reactions
Prof. Lutz F. TIETZE
12:50 Transportation to the City
15:00 Excursion
20:00 Conference Dinner (De Ark)
13/09/2008
Chairman
Dr. Kristof VAN EMELEN
09:00 π-Extended Tetrathiafulvalenes and Fullerenes: Complementary Topological and Electronic Molecules
Prof. Nazario MARTÍN
09:50 Synthesis of Natural Product Inspired Heterocyclic Compound Libraries
Prof. Floris RUTJES
10:20 Syntheses of Carbocyclic β-Amino Acids via Heterocyclic Intermediates
Prof. Ferenc FÜLOP
11:10 Coffee
Chairman
Prof. Erik VAN DER EYCKEN
11:40 Design and Synthesis of Novel Enzyme Inhibitors. Focus on Microwave-Acceleration and Metal-Catalyzed Transformations
Prof. Mats LARHED
12:30 Mn- and Fe-Catalyzed Coupling Reactions: Recent Advances
Prof. Gérard CAHIEZ
13:20 Annoucement of 24ECHC by Johannes Froehlich
13:30 Closing
13:40 Transportation to the City
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