EFMC 2nd Short Course on Medicinal Chemistry
11/04/2010
18:00Dinner
19:30Introduction to Safety & Attrition Workshop
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom)
21:00Close
12/04/2010
08:30General Overview of Current Safety and Toxicity Testing
Dr Dominic WILLIAMS
(UNIVERSITY OF LIVERPOOL, Liverpool, United Kingdom)
10:30Coffee Break
11:00Small Molecule Based Attrition (1) - Structural 'Alerts'
Dr Julian BLAGG
(THE INSTITUTE OF CANCER RESEARCH, Surrey, United Kingdom)
12:30Lunch
13:30Small Molecule Based Attrition (2) - Molecular Properties
Dr Julian BLAGG
(THE INSTITUTE OF CANCER RESEARCH, Surrey, United Kingdom)
15:30Tea Break
16:00Off-Target Based Attrition (1) - Ion Channel Safety
Dr Chris POLLARD
(ASTRAZENECA, Macclesfield, United Kingdom)
18:00Close
19:30Dinner
13/04/2010
08:30Off-Target Based Attrition (2) - Role of Transporter Interactions in Toxicology and Attrition
Dr Gerry KENNA
(ASTRAZENECA, Macclesfield, United Kingdom)
10:00Coffee Break
10:30Admet or DMPK Based Attrition
Dr Don WALKER
(PFIZER, Sandwich, United Kingdom)
12:30Lunch
13:30Choosing the Right Target
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom)
13:30Attrition (3) - Insilico Prediction Methods
Dr Alan STOBIE
(PFIZER, Sandwich, United Kingdom)
14:30The Safety and Attrition Game
18:00Close
19:30Dinner
14/04/2010
08:30Newer Methods of Predicting Toxicity (1) - Characterising Mechanisms of Toxicity
Dr Mark M. GOSINK
(PFIZER, Groton, United States)
10:00Coffee Break
10:30Newer Methods of Predicting Toxicity (2) - Use of Whole Cell Invitro Methods
Dr Jim DYKENS
(PFIZER, Sandwich, United Kingdom)
12:30Lunch
13:30Course Ends
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