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ASMC'11 St. Petersburg |
Confirmed Speakers |
| Metal-Catalyzed C–H Bond Functionalizations for Sustainable Synthesis |
Prof. Lutz ACKERMANN (GEORG-AUGUST UNIVERSITY GOETTINGEN, Goettingen, Germany) |
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| Chemical Probes for Epigenetics |
Dr Mark BUNNAGE (PFIZER, Boston, United States) |
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| Novel Metabotropic Glutamate Receptor 4 (mGluR4) Allosteric Potentiators for the Treatment of Parkinsons’s Disease |
Dr Sylvain CELANIRE (ADDEX PHARMACEUTICALS, Geneva, Switzerland) |
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| A few of my Favorite Rings: Catalysis Inspired by Lactones and Lactams |
Prof. Vy M. DONG (UNIVERSITY OF TORONTO, Toronto, Canada) |
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| Tofacitinib (CP-690,550): Discovery of a Potent and Selective JAK Inhibitor |
Dr Mark FLANAGAN (PFIZER, Connecticut, United States) |
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| Antibody Directed Cytotoxics |
Prof. John FLYGARE (GENENTECH, California, United States) |
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| From Homer to Hedgehog: Chemistry, Biological Investigations and Medical Perspectives of Cyclopamine |
Prof. Athanassios GIANNIS (UNIVERSITY OF LEIPZIG, Leipzig, Germany) |
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| Bicyclic Peptides with Tailored Binding Specificities for Therapeutic Application |
Prof. Christian HEINIS (ECOLE POLYTECHNIQUE FÉDÉRALE DE LAUSANNE (EPFL), Lausanne, Switzerland) |
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| Regioselective Reactions on a Chiral Substrate Controlled by the Configuration of a Chiral Catalyst |
Prof. Henri KAGAN (UNIVERSITY PARIS-SUD 11, ORSAY Cedex, France) |
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| Discovery and Development of Novel Antimalarials |
Dr Rodney KIP GUY (ST. JUDE CHILDREN'S RESEARCH HOSPITAL, Memphis, United States) |
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| Target Synthesis Directed Methodology Development |
Prof. Dawei MA (SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, Shanghai, China) |
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| Minor Enantiomer Recycling –
A Strategy for Improving Enantioselectivity
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Prof. Christina MOBERG (KTH SCHOOL OF CHEMICAL SCIENCE AND ENGINEERING, Stockholm, Sweden) |
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| Magical Power of d-Block Transition Metals—Pd-Catalyzed Cross-Coupling and Zr-Catalyzed Asymmetric carboalumination of Alkenes (ZACA) |
Prof. Ei-ichi NEGISHI (PURDUE UNIVERSITY, West Lafayette, United States) |
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| Maitotoxin. An Inspiration for Synthesis |
Prof. K.C. NICOLAOU (THE SCRIPPS RESEARCH INSTITUTE & UNIVERSITY OF CALIFORNIA, Houston, United States) |
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| Small Molecules Inhibitors of the WNT Signalling Pathway with Potential Applications in Oncology |
Dr Alessandro PADOVA (SIENA BIOTECH, Siena, Italy) |
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| Design Strategy for Preparation of Drug-like Polyheterocycles with Privileged Substructures for Discovery of Specific Small Molecule Modulators |
Prof. Seung Bum PARK (SEOUL NATIONAL UNIVERSITY, Seoul, Korea, South) |
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| Synthesis of Marine Polyketides as Promising Anticancer Agents |
Prof. Ian PATERSON (CAMBRIDGE UNIVERSITY, Cambridge, United Kingdom) |
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| GPR119: Knowledge Based Lead Identification |
Dr Sherrie L. PIETRANICO-COLE (ROCHE, NUTLEY NJ, United States) |
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| A Step Closer to Hepatitis C Remedy: TMC435, an HCV Protease Inhibitor in Advanced Clinical Trial |
Dr Pierre RABOISSON (JANSSEN PHARMACEUTICAL COMPANIES, Beerse, Belgium) |
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| The Many Uses of Noncovalent Mass Spectrometry in Early-stage Drug Discovery |
Dr Jean-Paul RENAUD (NOVALIX, Ostwald, France) |
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| The Resurgence of Covalent Drugs |
Dr Juswinder SINGH (AVILA THERAPEUTICS, United States) |
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| Lessons in Chemoselectivity: Total Synthesis of Polyphenolic Natural Products |
Prof. Scott SNYDER (COLUMBIA UNIVERSITY, New York, United States) |
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| Asymmetric Synthesis of Bioactive Molecules |
Prof. Mikiko SODEOKA (RIKEN, Hirosawa, Japan) |
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| Biochemical Efficiency, a Metrics for an Optimal Molecular Mechanism of Action |
Dr David SWINNEY (IRND3, Mountain View, United States) |
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| Drug Discovery by Programmed Self-Assembly |
Prof. Nicolas WINSSINGER (UNIVERSITY OF STRASBOURG, Geneva, Switzerland) |
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| Bromodomains a New Class of Epigenetic Targets Ripe for Small Molecule Drug Discovery |
Dr Jason WITHERINGTON (GLAXOSMITHKLINE R&D, Stevenage, United Kingdom) |
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| Validation of N-Myristoyltransferase as a Drug Target |
Prof. Paul WYATT (UNIVERSITY OF DUNDEE, Dundee, United Kingdom) |
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| Accelerated C-H Activation Reactions: Enantioselectivity and Positional Selectivity |
Prof Jin-Quan YU (THE SCRIPPS RESEARCH INSTITUTE, La Jolla, United States) |
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Selected Oral Communications |
| Small Molecule Inhibitors of the Neuropilin-1 VEGF-A Interaction |
Dr Philip FALLON (DOMAINEX, Saffron Walden, United Kingdom) |
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| Halogen Bonding in Protein–ligand Interactions |
Mr Leo HARDEGGER (ETH ZURICH, Zürich, Switzerland) |
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| The Chemical Biology Consortium-
and Experimental Therapeutics Program |
Dr Sanjay MALHOTRA (NATIONAL CANCER INSTITUTE, Frederick, United States) |
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| Adventures in Medicinal Chemistry and Knowledge Capture |
Dr Alexander MAYWEG (F. HOFFMANN-LA ROCHE LTD, BASEL, Switzerland) |
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| Identification of Bisaryloxy Azetidine Urea Derivatives as Fatty Acid Amide Hydrolase Inhibitors |
Dr Hans MEISSNER (VERNALIS, Winnersh, United Kingdom) |
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| Identification of Leads from the Tres Cantos Antimalarial Set: Cyclopropyl Carboxamides Show Good Oral Bioavailability and Efficacy In Malarial Animal Models |
Mrs Maria Lourdes RUEDA-BENEDE (GLAXOSMITHKLINE, Tres Cantos, Spain) |
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| Highly Efficient Catalytic System for C-H Activation: A Novel and Practical Synthesis of Angiotensin II Receptor Blockers |
Dr Masahiko SEKI (MITSUBISHI TANABE PHARMA CORPORATION, Fukuoka, Japan) |
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| The Grandisine Alkaloids as Selective δ-Opioid Receptor Agonists; When is a Natural Product not a Natural Product? |
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| Exploring the Rigid Mono- and Diamine Chemical Space |
Dr Dmytro VOLOCHNYUK (ENAMINE LTD., Kiev, Ukraine) |
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| Lead identification of a new class of P2Y12 inhibitors "From a low active and insoluble HTS hit to soluble and active lead compounds" |
Mr Fredrik ZETTERBERG (ASTRAZENECA, Gothenburg, Sweden) |
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| The Chemistry of Targeting Protein-Protein Interactions: Thinking Outdside of the Box |
Dr Giovanna ZINZALLA (LONDON SCHOOL OF PHARMACY, London, United Kingdom) |
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