Friday September 12, 2014 |
08:15 | Coffee/registration |
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09:00 | Welcome and opening |
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09:05 | Keynote lecture I |
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| Medicinal Chemistry Optimisation of Phenotypic Whole cell Screening Hits from SoftFocus Libraries |
Prof. Kelly CHIBALE (UNIVERSITY OF CAPE TOWN, Cape Town, South Africa) |
09:50 | YMCS competition presentation session I |
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| Session Chair: |
Dr Chris DE GRAAF (VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| A Chemical Probe for the CBP/P300 Bromodomains. Winner of the young medicinal chemist meeting in The United Kingdom |
Dr Duncan HAY (EVOTEC, Abingdon, United Kingdom) |
| Continuous Flow Chemistry as an Enabling Discovery Tool: Insights Into a Medchem and a Nutraceutical Application. Winner of the young medicinal chemist meeting in Italy |
Dr Lucia TAMBORINI (UNIVERSITÀ DI MILANO, Milano, Italy) |
| De Novo Structure-based Design of Novel Inhibitors of the Aspartic Protease Endothiapsin Exploiting Dynamic Combinatorial Chemistry |
Mr Milon MONDAL (, Groningen, The Netherlands) |
10:50 | Coffee break |
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11:15 | YMCS competition presentation session II |
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| Session Chair: |
Dr Rita GUEDES (UNIVERSITY OF LISBON, Lisbon, Portugal) |
| Straightforward Synthesis and Biological Evaluation of Sirna Prodrugs Partially Modified by Privaloyloxymethyl Groups. Winner of the young medicinal chemist meeting in France |
Mrs Christelle DUPOUY (UNIVERSITÉ DE MONTPELLIER, Montpellier, France) |
| Novel targeting of lipid signaling in aggressive breast cancer: A new therapeutic approach. Winner of the young medicinal chemist meeting in Israel |
Dr Nir BEN CHETRIT (WEIZMANN INSTITUTE OF SCIENCE, Rehovot, Israel) |
| Molecular mechanisms of functional selectivity of fenoterol derivatives towards the B2-Adrenergic Receptor. Winner of the young medicinal chemist meeting in Poland |
Mrs Karolina PAJAK (MEDICAL UNIVERSITY OF LUBLIN, Lublin, Poland) |
| De Novo Design of Lead-Like Chemical Entities for Kinase and GPCR Drug Targets |
Dr Tiago RODRIGUES (ETH ZÜRICH, Zürich, Switzerland) |
12:35 | Flash poster presentations |
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Dr Ewald EDINK (VU UNIVERSITY AMSTERDAM, Delft, The Netherlands) |
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Dr Stephanie GUERET (NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, Mölndal, Sweden) |
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Mr Rudi OLIVEIRA (IMED.ULISBOA, Lisboa, Portugal) |
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Ms Eleni KOTSAMPASAKOU (UNIVERSITY OF VIENNA, Vienna, Austria) |
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Mrs Sofia ALEXANDRE SANTOS (UNIVERSITY OF LISBON, Lisbon, Portugal) |
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Dr Ana RESSURREICAO (IMED.ULISBOA (INSTITUTO DE INVESTIGAÇÃO DO MEDICAMENTO), Lisboa, Portugal) |
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Mr Rafal URNIAZ (MEDICAL UNIVERSITY OF LUBLIN, Lublin, Poland) |
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Mrs Sara Cristina COVAS DA SILVA (UNIVERSITY OF LISBON, Lisboa, Portugal) |
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Ms Ramatoulie CAMARA (UNIVERSITY OF HERTFORDSHIRE, Hatfield, United Kingdom) |
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Mrs Mariana REIS (FACULTY OF PHARMACY -LISBON, Lisboa, Portugal) |
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Ms Daria GOLDMANN (UNIVERSITY OF VIENNA, Vienna, Austria) |
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Mr Carlos Jorge AZEVEDO COSTA RIBEIRO (INSTITUTO DE INVESTIGAÇÃO DO MEDICAMENTO (IMED.ULISBOA), Lisbon, Portugal) |
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Dr Andrea UNZUE (UNIVERSITY OF ZURICH, Zurich, Switzerland) Dr Agnese Chiara PIPPIONE (UNIVERSITY OF TURIN, Torino, Italy) |
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Dr Agnese Chiara PIPPIONE (UNIVERSITY OF TURIN, Torino, Italy) |
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Mr Pedro MIGUEL CAL (PHARMACY FACULTY - LISBON UNIVERSITY, Algés, Portugal) |
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Dr Frans SMIT (NORTH WEST UNIVERSITY - SOUTH AFRICA, Potchefstroom, South Africa) |
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Ms Nagore Isabel MARÍN RAMOS (COMPLUTENSE UNIVERSITY OF MADRID, Madrid, Spain) |
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Ms Marzena BARAN (JAGIELLONIAN UNIVERSITY MEDICAL COLLEGE, Krakow, Poland) |
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Dr Davide CARTA (UNIVERSITY OF PADOVA, Padova, Italy) |
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Ms Marta CARRASCO (FACULTY OF PHARMACY, UNIVERSITY OF LISBON, Lisbon, Portugal) |
13:05 | YMCS poster presentation session and lunch |
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14:50 | YMCS competition presentation session III |
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| Session Chair: |
Dr Fabrizio GIORDANETTO (TAROS CHEMICALS, New York, United States) |
| Functional Fragment Screening at GPCRS: Towards Signalling-Biased Fragments. Winner of the young medicinal chemist meeting in The Netherlands |
Dr Saskia NIJMEIJER (VU UNIVERSITY AMSTERDAM, AMSTERDAM, The Netherlands) |
| Maximizing the Performance of Consensus Scoring in Protein-Ligand Docking. Winner of the young medicinal chemist meeting in Greece |
Mr Thomas EVANGELIDIS (UNIVERSITY OF ATHENS, Athens, Greece) |
| Glycodendropeptides as a Potential Vaccine againsts Influenza A Virus. Winner of the young medicinal chemist meeting in Spain |
Dr Ainhoa MASCARAQUE (CSIC, Sevilla, Spain) |
| Optimising In Vivo Probes for the BET Bromodomains |
Ms Laura JENNINGS (UNIVERSITY OF OXFORD, Oxford, United Kingdom) |
| A Unified Approach for Rational Lead Discovery/Lead Optimization Toward Low Nanomolar Human Neutrophil Elastase Inhibitor Discovery |
Dr Susana DIAS LUCAS (INSTITUTO DE INVESTIGAÇÃO DO MEDICAMENTO (IMED.ULISBOA), Lisboa, Portugal) |
16:30 | Coffee break |
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16:55 | Keynote lecture II |
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| Keynote Speakers |
Dr Alexander V. MAYWEG (F. HOFFMANN-LA ROCHE LTD, Basel, Switzerland) |
17:40 | Closing and award ceremony |
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| Taros YMCS Presentation Prize |
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| Royal Society of Chemistry YMCS Poster Prize |
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| Roche YMCS Public's Choice Prize |
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18:00 | YMCS Networking and drinks |
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