|
Sunday April 12, 2015 |
18:00 | Dinner |
|
Monday April 13, 2015 |
| Breakfast (as of 7:30) |
|
08:30 | Introduction |
|
09:00 | Nuclear Receptor Protein-Protein Interactions |
Prof. Luc BRUNSVELD (EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands) |
10:30 | Coffee Break |
|
11:00 | Nuclear Receptor Protein-Protein Interactions - Part II |
Prof. Luc BRUNSVELD (EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands) |
12:30 | Lunch |
|
13:30 | Stabilization of PPIs: the Other Side of PPI Modulation |
Dr Christian OTTMANN (EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands) |
15:30 | Coffee Break |
|
16:00 | Stabilization of PPIs: the Other Side of PPI Modulation - Part II |
Dr Christian OTTMANN (EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands) |
17:30 | Day End |
|
Tuesday April 14, 2015 |
| Breakfast (as of 7:30) |
|
08:30 | Modern Methods for Targeting Low Affinity Protein-Protein Interactions: Structure and Function |
Prof. Anna MAPP (UNIVERSITY OF MICHIGAN, Ann-Arbor, United States) |
10:30 | Coffee Break |
|
11:00 | Modern Methods for Targeting Low Affinity Protein-Protein Interactions: Structure and Function - Part II |
Prof. Anna MAPP (UNIVERSITY OF MICHIGAN, Ann-Arbor, United States) |
12:30 | Lunch |
|
13:30 | Design and Synthesis of PPI-focussed Chemical Libraries |
Dr Fabrizio GIORDANETTO (TAROS CHEMICALS, New York, United States) |
15:30 | Coffee Break |
|
16:00 | Design and Evaluation of Biophysical Assays for the Identification of PPI-Modulators |
Dr Alexander WOLF (LEAD DISCOVERY, Dortmund, Germany) |
17:30 | Day End |
|
Wednesday April 15, 2015 |
| Breakfast (as of 7:30) |
|
08:30 | Developing Small Molecule Inhibitors of Bromodomain-Based Protein-Protein Interactions |
Prof. Stuart CONWAY (UNIVERSITY OF OXFORD, Oxford, United Kingdom) |
10:30 | Coffee Break |
|
11:00 | Structure-Based Guided Development & Experimental Validation of a Focused Chemical Library Dedicated to Orthosteric Modulation of Protein-Protein Interactions |
Dr Xavier MORELLI (CNRS, MARSEILLE CEDEX 9, France) |
12:30 | Wrap up and Lunch |
|
|