Online registration is still open! REGISTER NOW!
|
| Sunday July 3, 2016 |
| 14:00 | Registration |
|
| Session chair: |
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| 16:15 | Opening Ceremony |
Prof. Vinod SUBRAMANIAM
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands) |
| 16:30 | Opening Lecture - PL01 - How Natural Products Can Inspire Chemical Biology and Drug Discovery |
Prof. Herbert WALDMANN
(MAX PLANCK INSTITUTE OF MOLECULAR PHYSIOLOGY, Dortmund, Germany) |
| 17:15 | Welcome drink - sponsored by MDPI |
|
| Monday July 4, 2016 |
| Session chair: |
Dr Eelco RUIJTER
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| 09:00 | IL01 - Fluorinated Imaging Materials |
Prof. Tobias RITTER
(MAX-PLANCK-INSTITUT FÜR KOHLENFORSCHUNG, Mulheim, Germany) |
| 09:35 | PL02 - Organocatalytic Asymmetric Synthesis of Heterocycles |
Prof. Dieter ENDERS
(RWTH AACHEN, Aachen, Germany) |
| 10:20 | IL02 - The Development of Ligand Systems for Separating Minor Actinides from Lanthanides for Nuclear Fuel Reprocessing |
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom) |
| 10:55 | Coffee break and Exhibition |
|
| Session chair: |
Prof. Henk HIEMSTRA
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands) |
| 11:25 | IL03 - Stereoselective Heterocycle Synthesis Coupling Multicomponent Reactions with Biocatalysis or Organocatalysis |
Prof. Luca BANFI
(UNIVERSITY OF GENOA, Genova, Italy) |
| 12:00 | IL04 - Metal Free Cllick Reactions For Glycoconjugate Modification |
Prof. Geert-Jan BOONS
(THE UNIVERSITY OF GEORGIA, Athens, GA, United States) |
| 12:35 | IL05 - Target Family-Centric Privileged Structures: a Rich Playground for Diverse Heterocyclic Chemotypes |
Dr Gerhard MÜLLER
(MERCACHEM, Nijmegen, The Netherlands) |
| 13:10 | Lunch, Exhibition and Poster Session 1 (odd numbers) |
|
| Session chair: |
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom) |
| 14:40 | Elsevier presentation: Data-Driven Discovery: Deriving and Applying Actionable Information in Medicinal Chemistry |
|
| 15:00 | IL06 - Ynamides: Remarkable Building Blocks for Heterocyclic Synthesis |
Prof. Gwilherm EVANO
(ULB, Brussels, Belgium) |
| Heterocyclic Synthetic Methodology | Heterocyclic Synthetic Methodology | Medicinal Chemistry and Chemical Biology |
| Session chair: |
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom) |
|
| Session chair: |
Prof. Luca BANFI
(UNIVERSITY OF GENOA, Genova, Italy) |
|
| Session chair: |
Dr Alessia AMORE
(UBIQ, Amsterdam, The Netherlands) |
|
| 15:35 | KL01 - Alpha-Functionalization of Amines as a Tool for the Synthesis of Heterocycles and Natural Products
|
Prof. Till OPATZ
(JOHANNES GUTENBERG-UNIVERSITY, Mainz, Germany) |
|
| KL02 - First-in-Class MCRs Coupled with Cascade Reactions for the Generation of Molecular Complexity |
Prof. Christopher HULME
(UNIVERSITY OF ARIZONA, Tucson, United States) |
|
| KL03 - Biomimetic Natural Product Synthesis |
Dr Andrew LAWRENCE
(UNIVERSITY OF EDINBURGH, Edinburgh, United Kingdom) |
|
| 16:00 | OC01 - Poxim: A Novel N-Heterocyclic Carbene Equipped with Multifunctional Phosphine Oxide |
Prof. Yoichi HOSHIMOTO
(FACULTY OF ENGINEERING, OSAKA UNIVERSITY, Suita, Osaka, Japan) |
|
| OC06 - Asymmetric Synthesis of Natural Tetrahydroisoquinolines and Tetrahydroprotoberberines |
Dr Steen INGEMANN JORGENSEN
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC11 - Pyrazoloquinolinones, Revisited GABAA Receptor Tool Compounds
|
Mr David Chan Bodin SIEBERT
(TU WIEN, Wien, Austria) |
|
| 16:20 | OC02 - Efficient Approach to the Synthesis of 2,3-Substituted Furo[2,3-b]Pyridines
|
Mr Fernando FUMAGALLI
(UNIVERSITY OF SAO PAULO, Ribeirao Preto, Brazil) |
|
| OC07 - Synthesis of 3-Benzazepines by Metal-Free Oxidative C-H Bond Functionalization-Ring Expansion Tandem Reaction |
Mr Andrea GINI
(WISSENSCHAFTSZENTRUM STRAUBING, Straubing, Germany) |
|
| OC12 - Exploring Tryptophan Synthase as a Herbicidal Mode of Action |
Dr Matthew MCLACHLAN
(SYNGENTA, Bracknell, Berkshire, United Kingdom) |
|
| 16:40 | Coffee break and Exhibition |
|
|
|
|
| 17:10 | OC03 - Rapid Composition of Spiranoid Lactones: Access to Natural and Unexplored Frames
|
Dr Dmitry TSVELIKHOVSKY
(THE HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel) |
|
| OC08 - Combining Photochemistry and Catalysis: Rapid Access to SP3 - Rich Polyheterocycles from Simple Pyrroles |
Ms Emma BLACKHAM
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom) |
|
| OC13 - The Allylic Azide Rearrangement in Tandem with Huisgen Cycloaddition: Synthesis of Diverse Polyhydroxylated Nitrogen Containing Scaffolds |
Ms Rekha CHADDA
(SCHOOL OF CHEMISTRY, NUI GALWAY, Galway, Ireland) |
|
| 17:30 | OC04 - Nitrosoallenes: Reactivity and Applications to Heterocycles Synthesis
|
Dr Hiroki TANIMOTO
(NARA INSTITUTE OF SCIENCE AND TECHNOLOGY, Nara, Japan) |
|
| OC09 - Intramolecular Tsuji-Trost Cascade Cyclization as a Novel Synthetic Strategy Towards Muironolide A
|
Mr John BRAUN
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC14 - Synthesis and Potential Cytotoxic Activity of New Substituted Indazole Derivatives Bearing Pyrrole and 2-Pyrone
|
Mr Mohamed EL GHOZLANI
(UNIVERSTY SULTAN MY SLIMAN, Béni Mellal, Morocco) |
|
| 17:50 | OC05 - Synthesis of Highly and Diversely Substituted Heterocycles from Alk-3-yn-1-ones (Propargyl Ketones) |
Prof. Roman DEMBINSKI
(OAKLAND UNIVERSITY, Rochester, MI, United States) |
|
| OC10 - C-Brigded N-Heterocycles as New Ligands
|
Mr Tim-Daniel J. STUMPF
(JUSTUS-LIEBIG-UNIVERSITY GIESSEN, Giessen, Germany) |
|
| OC15 - Towards a Biomimetic Synthesis of Sciodole |
Mr Josh HOMER
(UNIVERSITY OF AUCKLAND, Auckland, New Zealand) |
|
|
| 18:10 | End of the day |
|
| Tuesday July 5, 2016 |
| Session Chair: |
Dr Tommi MEULEMANS
(MERCACHEM BV, Nijmegen, The Netherlands) |
| 09:00 | PL03 - Catalytic Approaches from the Synthesis of Enantiopure Biologically Relevant Heterocycles |
Prof. Floris RUTJES
(RADBOUD UNIVERSITY NIJMEGEN, Nijmegen, The Netherlands) |
| 09:45 | PL04 - Carbo- and Heterocycles via Metal-Catalyzed Cycloadditions |
Dr Fernando LOPEZ
(UNIVERSITY OF SANTIAGO DE COMPOSTELA (USC) AND SPANISH NATIONAL RESEARCH COUNCIL (CSIC), Santiago de Compostela, Spain) |
| 10:30 | IL07 - Photoactive Molecular and Supramolecular Materials Built-up with Heterocycles |
Prof. Gianluca M. FARINOLA
(UNIVERSITY OF BARI, Bari, Italy) |
| 11:05 | Coffee break and Exhibition |
|
| Session Chair: |
Prof. Huib OVAA
(NETHERLANDS CANCER INSTITUTE, Amsterdam , The Netherlands) |
| 11:30 | IL08 - Redesigning the Molecules of Nature: Lessons Learned from Total Synthesis |
Prof. Karl GADEMANN
(UNIVERSITY OF ZURICH, Zurich, Switzerland) |
| 12:05 | IL09 - Copper Catalysis for Synthesis of Enantiopure Alcohols, Amines and Heteroarenes |
Prof. Syuzanna HARUTYUNYAN
(UNIVERSITY OF GRONINGEN, Groningen, The Netherlands) |
| 12:40 | IL10 - C-H Functionalization for the Synthesis and Assembly of Heterocycles |
Prof. Lutz ACKERMANN
(GEORG-AUGUST UNIVERSITY GOETTINGEN, Goettingen, Germany) |
| 13:15 | Lunch, Exhibition and Poster Session 2 (even numbers) |
|
| Session Chair: |
Prof. Hermen OVERKLEEFT
(LEIDEN UNIVERSITY, Leiden, The Netherlands) |
| 14:45 | IL11 - Catalysis: A Versatile Tool for the Synthesis of Nitrogen-Containing Heterocycles |
Dr Geraldine MASSON
(INSTITUT DE CHIMIE DES SUBSTANCES NATURELLES CNRS, Gif-sur-Yvette, France) |
| Heterocyclic Synthetic Methodology | Heterocyclic Synthetic Methodology | Medicinal Chemistry and Chemical Biology |
| Session Chair: |
Prof. Hermen OVERKLEEFT
(LEIDEN UNIVERSITY, Leiden, The Netherlands) |
|
| Session Chair: |
Prof. Lutz ACKERMANN
(GEORG-AUGUST UNIVERSITY GOETTINGEN, Goettingen, Germany) |
|
| Session Chair: |
Prof. Henk TIMMERMAN
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
|
| 15:20 | KL04 - New Tricks for Old Heterocycles: from Natural Product Synthesis to Click-Like Functionalizations
|
Prof. Johan WINNE
(UNIVERSITEIT GENT, Ghent, Belgium) |
|
| KL05 - Synthesis of New Spiroacetals by Sustainable Gold Catalysis |
Prof. Norbert KRAUSE
(DORTMUND UNIVERSITY OF TECHNOLOGY, Dortmund, Germany) |
|
| KL06 - New Multicomponent Reactions and Strategies to Heterocyclic and Macrocyclic Peptides |
Dr Daniel GARCÍA RIVERA
(LEIBNIZ INSTITUTE OF PLANT BIOCHEMISTRY / UNIVERSITY OF HAVANA, La Habana, Cuba) |
|
| 15:45 | OC16 - Synthesis of Highly Enantioenriched Pyrrolo[1,2-a]Quinolines. Organocatalyzed Domino Cyclopropane Ring Opening/aza-Michael/aldol Reaction Followed by Acid-Promoted Lactamization
|
Mr Eduardo SANCHEZ
(UPV/EHU UNIVERSITY OF THE BASQUE COUNTRY, Leioa, Spain) |
|
| OC21 - Is Gold Catalysis a Competitive Method toward Heterocycles ?
|
Mrs Solène MIASKIEWICZ
(STRASBOURG UNIVERSITY, Strasbourg, France) |
|
| OC26 - Palladium-Catalyzed Isocyanide Insertion in Construction of Diverse Heterocycles
|
Dr Esther VICENTE GARCIA
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands) |
|
| 16:05 | OC17 - Brönsted-Acid Catalysed C2-Alkenylation of Aromatic Nitrogen Heterocycles |
Mr Giacomo CRISENZA
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom) |
|
| OC22 - Aliphatic N-Heterocycle Synthesis through Direct C-H Bond Amination
|
Mr Petrus KUIJPERS
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC27 - Biologically Active Indolines - Novel Multi-Functional Indolinic Drugs for the Treatment of Inflammatory Diseases
|
Prof. Abraham NUDELMAN
(BAR ILAN UNIVERSITY, Ramat Gan, Israel) |
|
| 16:25 | Coffee break and Exhibition |
|
|
|
|
| 17:00 | OC18 - Rearrangement and Cycloaddition Reactions of Donor-Acceptor Cyclopropanes
|
Prof. Daniel B. WERZ
(TU BRAUNSCHWEIG, Braunschweig, Germany) |
|
| OC23 - 3-Diazoindolin-2-Imines: A Novel Class of Metal Carbene Precursors for the Syntheses of Indole Derivatives
|
Prof. Yanguang WANG
(ZHEJIANG UNIVERSITY, Hangzhou, China) |
|
| OC28 - Asymmetric Reduction of Enamines towards the Synthesis of (-)-Cytisine and Heterocyclic Building Blocks
|
Mr Hugo REGO CAMPELLO
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom) |
|
| 17:20 | OC19 - Pd- and Cu-Catalyzed Stereo- and Regiocontrolled Decarboxylative / C-H Alkenylation of Heroarenes |
Dr Cedric SCHNEIDER
(UNIVERSITY OF ROUEN, Mont Saint Aignan, France) |
|
| OC24 - Donor-Acceptor Cyclopropanes in Synthesis of Azaheterocycles
|
Prof. Igor TRUSHKOV
(M V LOMONOSOV MOSCOW STATE UNIVERSITY, Moscow, Russia) |
|
| OC29 - Biology-Oriented Synthesis Based on Privileged Structures: Building Framework Diversity Around Pyrrole Cores |
Prof. José Carlos MENÉNDEZ
(UNIVERSIDAD COMPLUTENSE, Madrid, Spain) |
|
| 17:40 | OC20 - Enantioselective Organocatalyzed Α-Sulfanylation of Isoxazolidin-5-ones: An Approach To b2,2-Amino Acids
|
Mr Timothée CADART
(LABORATOIRE COBRA UMR 6014, ROUEN, France) |
|
| OC25 - Chirality in Boron-Chelated Dipyrromethene Fluorophores: Synthesis and Chiroptical Investigations |
Dr Michael HALL
(NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom) |
|
| OC30 - Exploring the Antifungal and Antibiofilm Properties of Imidazolium Salts and Fluorescent Benzannulated Benzimidazoles |
Prof. Henri SCHREKKER
(UNIVERSIDADE FEDERAL DO RIO GRANDE DO SUL, Porto Alegre-RS, Brazil) |
|
|
| 18:00 | End of the day |
|
| 18:30 | Boat tour and Conference dinner |
|
| Wednesday July 6, 2016 |
| Session Chair: |
Prof. Karl Anker JOERGENSEN
(AARHUS UNIVERSITY, Aarhus, Denmark) |
| 09:00 | IL12 - Complex Natural Product as a Driving Force for Discovery in Organic Synthesis and Chemical Biology |
Prof. Xiaoguang LEI
(PEKING UNIVERSITY, Beijing, China) |
| 09:35 | IL13 - Metallation–Substitution of Saturated Nitrogen Heterocycles |
Prof. Iain COLDHAM
(UNIVERSITY OF SHEFFIELD, Sheffield, United Kingdom) |
| 10:10 | PL05 - Springer Junior Heterocyclic Chemistry Award Lecture (chaired by Bert Maes, editor of Springer)
Exploiting the Reactivity of Strained Rings and Hypervalent Bonds for the Synthesis of Heterocycles |
Prof. Jerome WASER
(LABORATORY OF CATALYSIS AND ORGANIC SYNTHESIS, EPFL, Lausanne, Switzerland) |
| 10:55 | IL14 - α-Perluoroalkylated Cyclic Imines as a Valuable Building Blocks
|
Prof. Dr Valentine G. NENAJDENKO
(MOSCOW STATE UNIVERSITY, Moscow, Russia) |
| 11:30 | Coffee break and Exhibition |
|
| Session Chair: |
Prof. Floris RUTJES
(RADBOUD UNIVERSITY NIJMEGEN, Nijmegen, The Netherlands) |
| 11:55 | IL15 - New Strategies for the Synthesis of Heterocyclic through Multicomponent Reactions and Metal-Catalyzed Isomerization |
Prof. Thomas NIELSEN
(NOVO NORDISK, Copenhagen N, Denmark) |
| 12:30 | PL06 - Making Molecular Prosthetics with a Small Molecule Synthesizer |
Prof. Martin D. BURKE
(UNIVERSITY OF ILLINOIS, Urbana, United States) |
| 13:15 | Lunch |
|
| Heterocyclic Synthetic Methodology | Enabling Technologies | Medicinal Chemistry and Chemical Biology |
| Session Chair: |
Prof. Martin D. BURKE
(UNIVERSITY OF ILLINOIS, Urbana, United States) |
|
| Session Chair: |
Dr Maikel WIJTMANS
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
|
| Session Chair: |
Prof. Rob LEURS
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
|
| 14:15 | KL07 - Gamma-Alkylidenebutenolides and Gamma-Hydroxybutyrolactams: Preparation and Reactivity |
Dr Laurent COMMEIRAS
(AIX-MARSEILLE UNIVERSITY, Marseille cedex 20, France) |
|
| KL08 - Functionalization of Heterocycles via C–H Activation and Photoredox Catalysis in Batch and Continuous Flow
|
Dr Timothy NOEL
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands) |
|
| KL09 - Going Beyond ß-Amino Acid Derivatives as Inhibitors of Cathepsin A |
Dr Sven RUF
(SANOFI-AVENTIS DEUTSCHLAND GMBH, Frankfurt am Main, Germany) |
|
| 14:40 | OC31 - Picolinic Acid Ligand-Promoted Palladium-Catalyzed C-H Acetoxylation of Simple Arenes |
Dr M. Angeles FERNANDEZ-IBANEZ
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC36 - N-Heterocyclic Carbene Ligands in Iridium Complexes for the Detection of Pyridine Analogues in NMR by Non-Hydrogenative Para-Hydrogen Induced Hyperpolarization |
Dr Martin FEITERS
(RADBOUD UNIVERSITY, Nijmegen, The Netherlands) |
|
| OC41 - Designing Residence Time into Heterocyclic Ligands for Drug Targets
|
Dr Julien LOUVEL
(LACDR, Leiden, The Netherlands) |
|
| 15:00 | OC32 - Stereoselective Transformations of 2h-Chromene Derivatives |
Prof. Tibor KURTÁN
(UNIVERSITY OF DEBRECEN, Debrecen, Hungary) |
|
| OC37 - Expansion of the Concept of Nonlinear Effects in Catalytic Reactions Beyond Asymmetric Catalysis
|
Prof. Michael SCHNÜRCH
(TU WIEN, Wien, Austria) |
|
| OC42 - Photopharmacology |
Mr Mickel HANSEN
(RIJKSUNIVERSITEIT GRONINGEN, Groningen, The Netherlands) |
|
| 15:20 | Coffee break and Exhibition |
|
|
|
|
| 15:50 | OC33 - Scope and Limitations of the Organocatalyzed Domino Vinylogous Aldol Oxa Michael Reaction |
Ms Larissa GEIGER
(KARLSRUHE INSTITUTE OF TECHNOLOGY, Karlsruhe, Germany) |
|
| OC38 - Direct Heteroatom Incorporating Ester to Arene Transformation: Modular Synthesis of Fluorescent Dyes
|
Mr Christian FISCHER
(UNIVERSITY OF BASEL, Basel, Switzerland) |
|
| OC43 - Novel Synthesis of Tetrahydroisoquinoline Derivatives Using Petasis Reaction |
Dr Agnieszka GRAJEWSKA
(ADAM MICKIEWICZ UNIVERSITY, Poznan, Poland) |
|
| 16:10 | OC34 - Dearomative Arylation of Electrophilic Indoles for the Total Synthesis of Natural Products |
Prof. Guillaume VINCENT
(UNIVERSITÉ PARIS SUD INSTITUT DE CHIMIE MOLÉCULAIRE ET DES MATÉRIAUX D'ORSAY (ICMMO), Orsay, France) |
|
| OC39 - Methodology Development Towards the Lasso Peptide Series |
Prof. Jan VAN MAARSEVEEN
(UNIVERSITEIT VAN AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC44 - Palladium Catalyzed C-Arylation of Amino Acid Derived Hydantoins
|
Mr Josep MAS ROSELLO
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom) |
|
| 16:30 | OC35 - Integrative Methodology for Iterative Theory-Experiment Driven Multicomponent Reaction Development |
Mr Art KRUITHOF
(VU AMSTERDAM, Amsterdam, The Netherlands) |
|
| OC40 - A Lab-Scale Reactor for the Continuous Generation of Anhydrous Diazomethane |
Dr Doris DALLINGER
(UNIVERSITY OF GRAZ, Graz, Austria) |
|
| OC45 - Enantioselective Synthesis of 4-Arylpyridine Atropisomers by Central-to-Axial Chirality Conversion
|
Ms Ophélie QUINONERO
(ISM2 - INSTITUT DES SCIENCES MOLÉCULAIRE DE MARSEILLE, Marseille, France) |
|
|
| Session Chair: |
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| 16:50 | PL07 - Organocatalysis for Diversity-Oriented Synthesis |
Prof. Karl Anker JOERGENSEN
(AARHUS UNIVERSITY, Aarhus, Denmark) |
| 17:35 | Poster prizes |
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| 17:50 | End of the Symposium |
|
|
