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| Sunday April 24, 2016 |
| 18:00 | Dinner |
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| 20:00 | Opening |
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| 20:15 | Basic Principles of Enzymology |
Dr Laurie LEBRUN
(CELGENE, San Diego, United States) |
| Monday April 25, 2016 |
| 07:30 | Breakfast |
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| 08:30 | Introduction |
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| 09:00 | Protein Kinase Inhibitors |
Dr Gerhard MÜLLER
(MERCACHEM, Nijmegen, The Netherlands) |
| 10:30 | Coffee Break |
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| 11:00 | Epigenetic Target Families in Medicinal Chemistry |
Prof. Paul BRENNAN
(UNIVERSITY OF OXFORD, Oxford, United Kingdom) |
| 12:30 | Lunch |
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| 13:30 | BETting on Epigenetic Targets: From Phenotypic Discovery to First Time in Man |
Dr Chun-wa CHUNG
(GLAXOSMITHKLINE R&D, Stevenage, United Kingdom) |
| 15:00 | Coffee Break |
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| 15:30 | Hands on Tutorial - Case Study I: Development of a Kinase Inhibitor |
Dr Leon VAN BERKOM (MERCACHEM, Nijmegen, The Netherlands)
Dr Toine VAN DEN BERGH (MERCACHEM, Nijmegen, The Netherlands) |
| 18:00 | Day End |
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| Tuesday April 26, 2016 |
| 07:30 | Breakfast |
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| 08:30 | Proteases as Drug Targets |
Dr Holger SELLNER
(NOVARTIS PHARMA AG, Basel, Switzerland) |
| 10:00 | Coffee Break |
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| 10:30 | Proteasome Inhibitors |
Prof. Michael GROLL
(TECHNISCHE UNIVERSITÄT MÜNCHEN, Garching, Germany) |
| 12:00 | Lunch |
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| 13:00 | Glycomimetics - an Underexplored Compound Class for Medicinal Chemistry |
Prof. Dr Beat ERNST
(UNIVERSITY OF BASEL, Basel, Switzerland) |
| 14:30 | Coffee Break |
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| 15:00 | Hands on Tutorial - Case Study II: Development of a HIV Medicine |
Dr Stijn GREMMEN (MERCACHEM, Nijmegen, The Netherlands)
Dr Harald ALBERS (MERCACHEM, Nijmegen, The Netherlands) |
| 17:30 | Day End |
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| Wednesday April 27, 2016 |
| 07:30 | Breakfast |
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| 08:30 | The PDE Family and Inhibitors |
Dr Andrew BELL
(IMPERIAL COLLEGE LONDON, London, United Kingdom) |
| 10:00 | Coffee break |
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| 10:30 | Fragment-Based Lead Generation |
Prof. Iwan DE ESCH
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands) |
| 12:30 | Wrap-up and Lunch |
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