MedChem 2007 - New Drugs and Drug Candidates:
Recent Achievements in Medicinal Chemistry
26/10/2007
08:00Registration
08:50Introduction
09:00Nexavar - A Novel Inhibitor of Signal Transduction
Dr Bernd RIEDL
(BAYER PHARMA, Wuppertal, Germany)
09:50Design, Synthesis and Biological Activity of Therapeutics Targeting the PI3K Pathway
Dr. Carlos GARCIA-ECHEVERRIA
(NOVARTIS PHARMA, Basel, Switzerland)
10:40Coffee-break & poster session
11:10Discovery of Sitagliptin and Other Novel DPP4 Inhibitors
Dr Tesfaye BIFTU
(MERCK, Rahway, United States)
12:00Hit-to-lead studies on Aminopropoxy phenyloxazolines. Discovery of a novel class of potent H3R ligands for the treatment of cognitive dysfunction

(EYEDPHARMA)
12:20Sandwich lunch & posters
13:40Dual NK3/NK1 Receptor Antagonism: A Novel Approach for the Treatment of Psychotic Disorders
Dr. Patrick SCHNIDER
(F. HOFFMANN-LA ROCHE, Basel, Switzerland)
14:30Isoindolinones as promising inhibitors of the MDM2-P53 protein-protein interaction
Dr. Eric VALEUR
(MERCK SERONO, Chilly Mazarin, France)
14:50ETHR inhibitors as TB drug boosters: A new strategy to fight tuberculosis
Prof. Nicolas WILLAND
(UNIVERSITY OF LILLE, Lille, France)
15:10Coffee-break & poster session
15:40Discovery of R256918 a Gut-Selective MTP Inhibitor to Treat Obesity
Dr Lieven MEERPOEL
(JOHNSON & JOHNSON PRD, Beerse, Belgium)
16:30Inhibitors of Thrombin Activatable Fibrinolysis Inhibitor (TAFIa)
Dr Mark BUNNAGE
(PFIZER, Boston, United States)
17:20Closing remarks
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